Konstantin S. Chunikhin

1-Tosyl-2-trifluoroacetylindole as Promising Partner for Synthesis of Fused Fluorinated Heterocycles

Konstantin S. Chunikhin · Chemical Science International Journal · 2019

We prepared 1-tosyl-2-trifluoroacetylindole - a novel example of an electron-deficient indole with an electrophilic C(3) position. This substance was involved in cyclocondensation with a variety of amidines to propose a new general pathway to 8H-[4,5-b]indolopyrimidines with yiel...