Skip to content
Research Article Open access CC BY 4.0

Optimization of Synthesis Process of 4-Methylquinazoline

Juan Liu, Yun Yang, Liangchun Li

International Research Journal of Pure and Applied Chemistry · pp. 1–5 · Published 21 Aug 2017

10.9734/IRJPAC/2017/35918

Abstract

4-Methylquinazoline was synthesized with 2-aminoacetophenone and formamide as the starting materials. The reaction conditions, including catalyst, ratio of substrates, temperature and time were optimized. Results showed that the optimal condition were as follows: Catalyst BF3-Et2O, the molar ratio of 2-aminoacetophenone: BF3-Et2O = 1:0.5, the weight ratio of 2-aminoacetophenone: formamide = 1:52, temperature 150°C, and time 6 h. Under the optimal conditions, the yield of the reaction achieved the highest (86%), which are better than the past reports.

Quinazolines 4-methylquinazoline synthesis Lewis acid reaction condition

Cited by 1

Copper-catalyzed oxidative amination of methanol to access quinazolines

Gandhesiri Satish, Ashok Polu, Laxman Kota · Organic & Biomolecular Chemistry · 2019

Article metrics

Real usage data collected on this platform.

0

Page views

0

PDF downloads

0

Outbound clicks

1

Citations

Views by country

Approximate, from request IP at view time — not citizenship or institution. Countries with fewer than 5 views are grouped as "Other".

No views recorded yet.

Traffic sources

Referring site, by host.

No traffic recorded yet.

Views and downloads exclude known bots/crawlers. Citations combines this platform's own DOI-resolved index with each external source's own reported total — see Cited by above for individually listed citing works. Last refreshed 0 seconds ago.