Synthesis, Antiviral and Kinesin Eg5 Activities of New Indomethacin Analogues

References (44)

1. 1 Isolation of a T-Lymphotropic Retrovirus from a Patient at Risk for Acquired Immune Deficiency Syndrome (AIDS) [DOI]
2. 2 Detection, Isolation, and Continuous Production of Cytopathic Retroviruses (HTLV-III) from Patients with AIDS and Pre-AIDS [DOI]
3. 3 3'-Azido-3'-deoxythymidine (BW A509U): an antiviral agent that inhibits the infectivity and cytopathic effect of human T-lymphotropic virus type III/lymphadenopathy-associated virus in vitro. [DOI]
4. 4 Small Molecule Inhibitor of Mitotic Spindle Bipolarity Identified in a Phenotype-Based Screen [DOI]
5. 5 Nonsteroidal Anti-inflammatory Drugs as Anticancer Agents: Mechanistic, Pharmacologic, and Clinical Issues [DOI]
6. 6 Differential inhibition of prostaglandin endoperoxide synthase (cyclooxygenase) isozymes by aspirin and other non-steroidal anti-inflammatory drugs. [DOI]
7. 7 Gradient selection in inverse heteronuclear correlation spectroscopy [DOI]
8. 8 Indomethacin and Aspirin abolish Prostaglandin Release from the Spleen [DOI]
9. 9 Pharmacological analysis of cyclooxygenase-1 in inflammation [DOI]
10. 10 Microtubule motors in mitosis [DOI]
11. 11 Structural and Functional Basis of Cyclooxygenase Inhibition [DOI]
12. 12 Microtubule-targeted anticancer agents and apoptosis [DOI]
13. 13 Experiments for recording pure-absorption heteronuclear correlation spectra using pulsed field gradients [DOI]
14. 14 Tetrazolium-based colorimetric assay for the detection of HIV replication inhibitors: revisited 20 years later [DOI]
15. 15 In Search of a Novel Anti-HIV Drug: Multidisciplinary Coordination in the Discovery of 4-[[4-[[4-[(1 E )-2-Cyanoethenyl]-2,6-dimethylphenyl]amino]-2- pyrimidinyl]amino]benzonitrile (R278474, Rilpivirine) [DOI]
16. 16 Evidence that Monastrol Is an Allosteric Inhibitor of the Mitotic Kinesin Eg5 [DOI]
17. 17 New Palladium Carbene Catalysts for the Heck Reaction of Aryl Chlorides in Ionic Liquids [DOI]
18. 18 Cyclooxygenase-2 Biology [DOI]
19. 19 Indomethacin: A New Non-steroid Anti-inflammatory Agent [DOI]
20. 20 Indomethacin Has a Potent Antiviral Activity against Sars Coronavirus [DOI]
21. 21 A replicon-based bioassay for the measurement of interferons in patients with chronic hepatitis C [DOI]
22. 22 Novel non-nucleoside inhibitors of HIV-1 reverse transcriptase. 1. Tricyclic pyridobenzo- and dipyridodiazepinones [DOI]
23. 23 Role of endothelial adhesion molecules in NSAID-induced gastric mucosal injury [DOI]
24. 24 A microassay for ATPase [DOI]
25. 25 The Activity of Plant-Derived Antiretroviral Proteins MAP30 and GAP31 against Herpes Simplex Virus Infectionin Vitro [DOI]
26. 26 ATPase Mechanism of Eg5 in the Absence of Microtubules: Insight into Microtubule Activation and Allosteric Inhibition by Monastrol [DOI]
27. 27 Indolyl esters and amides related to indomethacin are selective COX-2 inhibitors [DOI]
28. 28 Respiratory Syncytial Virus (RSV) Infection Induces Cyclooxygenase 2: A Potential Target for RSV Therapy [DOI]
29. 29 The 2′-Trifluoromethyl Analogue of Indomethacin Is a Potent and Selective COX-2 Inhibitor [DOI]
30. 30 NSAIDs: Old Drugs Reveal New Anticancer Targets [DOI]
31. 31 Type C Virus-Producing Cell Lines Derived from Adult T Cell Leukemia [DOI]
32. 32 Novel mechanism of resistance to paclitaxel (Taxol) in human K562 leukemia cells by combined selection with PSC 833.
33. 33 Molecular Basis of the Time-Dependent Inhibition of Cyclooxygenases by Indomethacin [DOI]
34. 34 Pathway of ATP Hydrolysis by Monomeric Kinesin Eg5 [DOI]
35. 35 COX inhibitors Indomethacin and Sulindac derivatives as antiproliferative agents: Synthesis, biological evaluation, and mechanism investigation [DOI]
36. 36 Tenidap, a structurally novel drug for the treatment of arthritis: Antiinflammatory and analgesic properties [DOI]
37. 37 Utility of MetaSite in Improving Metabolic Stability of the Neutral Indomethacin Amide Derivative and Selective Cyclooxygenase-2 Inhibitor 2-(1-(4-Chlorobenzoyl)-5-methoxy-2-methyl-1H-indol-3-yl)-N-phenethyl-acetamide [DOI]
38. 38 Synthesis, structural characterization and cytotoxic activity of organotin derivatives of indomethacin [DOI]
39. 39 Synthesis and biological evaluation of indomethacin analogs possessing a N-difluoromethyl-1,2-dihydropyrid-2-one ring system: A search for novel cyclooxygenase and lipoxygenase inhibitors [DOI]
40. 40 Desmethyl Derivatives of Indomethacin and Sulindac as Probes for Cyclooxygenase-Dependent Biology [DOI]
41. 41 1H- and 13C-NMR Study of Some 6,7-Dihaloquinolone Nucleosides and Their Derivatives [DOI]
42. 42 Cytostatic and Antiviral Activity Evaluations of Hydroxamic Derivatives of Some Non‐steroidal Anti‐inflammatory Drugs [DOI]
43. 43 Indomethacin inhibits viral RNA and protein synthesis in cells infected with vesicular stomatitis virus [DOI]
44. 44 ChemInform Abstract: Novel Non‐Nucleoside Inhibitors of HIV‐1 Reverse Transcriptase. Part 1. Tricyclic Pyridobenzo‐ and Dipyridodiazepinones. [DOI]

Cited by 0

No indexed citations yet.

Related research

• Antimicrobial Profile of Selected Snake Venoms and Their Associated Enzymatic Activities — shares topic coverage
• In vitro Antiviral Activity of Nauclea latifolia Root Bark Extract Against the Respiratory Syncytial Virus — shares topic coverage
• Review on Ethno-botany, Virucidal Activity, Phytochemistry and Toxicology of Solanum genus: Potential Bio-resources for the Therapeutic Management of Covid-19 — shares topic coverage
• Aloe vera (L.) Burm. F. as a Potential Anti-COVID-19 Plant: A Mini-review of Its Antiviral Activity — shares topic coverage
• Antiviral Activity of Approved Anti-Inflammatory Drugs and Prospects for Drug Repurposing: A review — shares topic coverage